Gianluca Papeo

Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1<i>H</i>-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy

Gianluca Papeo, Helena Posteri, Daniela Borghi et al. · Journal of Medicinal Chemistry · 2015 · 139 citations · Full text

Cancer Therapy, Drug Target, Pharmacotherapy +18

Oxindole alkaloids. A novel non-biomimetic entry to (−)-Horsfiline.

Giovanni Palmisano, Rita Annunziata, Gianluca Papeo et al. · Tetrahedron Asymmetry · 1996 · 94 citations

Bioorganic Chemistry, Biochemistry, Medicine +6

Sensitivity Improvement in ¹⁹F NMR-Based Screening Experiments:  Theoretical Considerations and Experimental Applications

Claudio Dalvit, Nicola Mongelli, Gianluca Papeo et al. · Journal of the American Chemical Society · 2005 · 63 citations

A Straightforward Total Synthesis of (−)‐Chaetominine

Beatrice Malgesini, Barbara Forte, Daniela Borghi et al. · Chemistry - A European Journal · 2009 · 47 citations

Straightforward Total Synthesis, Bioorganic Chemistry, Indole Ring +10

Polyfluorinated Amino Acids for Sensitive ¹⁹F NMR-Based Screening and Kinetic Measurements

Gianluca Papeo, Patrizia Giordano, Maria Gabriella Brasca et al. · Journal of the American Chemical Society · 2007 · 47 citations

Small Arginine-containing Peptides, Amino Acids, Peptide Engineering +19