Gianluca Papeo - Concepedia

Author

Gianluca Papeo

Nerviano Medical Sciences ORCID

Also Known As

G Papeo, G. PAPEO, G. Papeo, Gianluca Papeo

Publications

1.2K

Citations

H-Index

Concepts

All Affiliations

Nerviano Medical Sciences University of Milan Université de Montréal

About

Gianluca Papeo is an author at Nerviano Medical Sciences specializing in natural sciences, organic chemistry, and biochemistry.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Natural Sciences	10	10	468
2	Biochemistry	9	9	427
3	Medicine	7	7	386
4	Biomolecular Engineering	5	5	135
5	Engineering	4	4	87

Gianluca Papeo

Publications

766

Citations

H-Index

Page 1

	Year	Citations
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1<i>H</i>-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy Gianluca Papeo, Helena Posteri, Daniela Borghi, Journal of Medicinal Chemistry Cancer TherapyDrug TargetPharmacotherapyParp-1 Selective InhibitorChemical Biology	2015	139
Oxindole alkaloids. A novel non-biomimetic entry to (−)-Horsfiline. Giovanni Palmisano, Rita Annunziata, Gianluca Papeo, Tetrahedron Asymmetry Bioorganic ChemistryBiochemistryMedicineNatural SciencesSecondary Metabolite	1996	94
Sensitivity Improvement in <sup>19</sup>F NMR-Based Screening Experiments: Theoretical Considerations and Experimental Applications Claudio Dalvit, Nicola Mongelli, Gianluca Papeo, Journal of the American Chemical Society	2005	63
A Straightforward Total Synthesis of (−)‐Chaetominine Beatrice Malgesini, Barbara Forte, Daniela Borghi, Chemistry - A European Journal Straightforward Total SynthesisBioorganic ChemistryIndole RingHeterocyclicNatural Sciences	2009	47
Polyfluorinated Amino Acids for Sensitive <sup>19</sup>F NMR-Based Screening and Kinetic Measurements Gianluca Papeo, Patrizia Giordano, Maria Gabriella Brasca, Journal of the American Chemical Society Small Arginine-containing PeptidesAmino AcidsPeptide EngineeringMolecular BiologyPeptide Science	2007	47
Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515 Gianluca Papeo, Paolo Orsini, Nilla Avanzi, ACS Medicinal Chemistry Letters	2019	42
Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases Francesco Casuscelli, Elena Ardini, Nilla Avanzi, Bioorganic & Medicinal Chemistry Medicinal ChemistryPim KinasesBiochemistryMedicineNatural Sciences	2013	36
Total synthesis of (±)-cyclooroidin Gianluca Papeo, María Antonia Gómez-Zurita Frau, Daniela Borghi, Tetrahedron Letters PharmacologyOrganic ChemistryNatural Product SynthesisTotal Synthesis	2005	33
Synthesis of 3<sub>10</sub>-Helix-Inducing Constrained Analogues of <scp>l</scp>-Proline Stephen Hanessian, Gianluca Papeo, Kamal Fettis, The Journal of Organic Chemistry	2004	32
Synthesis of 7,5-fused bicyclic lactams by stereoselective radical cyclization Lino Colombo, Marcello Di Giacomo, Gianluca Papeo, Tetrahedron Letters Organic Chemistry7,5-Fused Bicyclic LactamsStereoselective SynthesisChemistrySynthetic Chemistry	1994	31

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