David P. Temelkoff

Carbamoyl Pyridone HIV-1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)

Brian A. Johns, Takashi Kawasuji, Jason G. Weatherhead et al. · Journal of Medicinal Chemistry · 2013 · 181 citations · Full text

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +15

Structural Basis for Inhibitor-Induced Aggregation of HIV Integrase

Kushol Gupta, Vesa Turkki, Scott Sherrill-Mix et al. · PLoS Biology · 2016 · 66 citations · Full text

Amino Acids, Protein Assembly, Hiv Integrase +17

N-Glycoside neoglycotrimers from 2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl azide

David P. Temelkoff, Mat­thias Zeller, Peter Norris · Carbohydrate Research · 2006 · 36 citations

N-glycoside Neoglycotrimers, Bioorganic Chemistry, Biochemistry +4

Rapid Access to Glucopyranosyl-1,2,3- triazoles via Cu(I)-catalyzed Reactions in Water

Peter Norris, Rakesh A. Akula, David P. Temelkoff et al. · Heterocycles · 2004 · 29 citations · Full text

Rapid Access, Engineering, Organic Chemistry +16

The design of 8-hydroxyquinoline tetracyclic lactams as HIV-1 integrase strand transfer inhibitors

Emile J. Velthuisen, Brian A. Johns, David P. Temelkoff et al. · European Journal of Medicinal Chemistry · 2016 · 25 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +10