Huangshu Lei

Identification of NVP-TNKS656: The Use of Structure–Efficiency Relationships To Generate a Highly Potent, Selective, and Orally Active Tankyrase Inhibitor

Michael D. Shultz, Atwood K. Cheung, C.A. Kirby et al. · Journal of Medicinal Chemistry · 2013 · 122 citations · Full text

Drug Target, Selective Tankyrase Inhibitors, Pharmacotherapy +18

1-Amino-4-benzylphthalazines as Orally Bioavailable Smoothened Antagonists with Antitumor Activity

Karen Miller‐Moslin, Stefan Peukert, Rishi K. Jain et al. · Journal of Medicinal Chemistry · 2009 · 106 citations · Full text

Pharmaceutical Science, Antitumor Activity, Pharmacotherapy +16

Optimization of 4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine IGF-1R tyrosine kinase inhibitors towards JNK selectivity

Stanley D. Chamberlain, Anikó M. Redman, Joseph W. Wilson et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 57 citations · Full text

Medicinal Chemistry, Biochemistry, Natural Sciences +8

Design, synthesis, and biological evaluation of dihydroartemisinin–fluoroquinolone conjugates as a novel type of potential antitubercular agents

Fu-Wei Zhou, Huangshu Lei, Fan Li et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 51 citations

Bioorganic Chemistry, Novel Type, Biochemistry +9

Synthesis of Phytyl- and Chroman-Derivatized Photoaffinity Labels Based on α-Tocopherol

Huangshu Lei, Jeffrey Atkinson · The Journal of Organic Chemistry · 2000 · 37 citations