Stéphane Sautet

Identification of 1,5-Naphthyridine Derivatives as a Novel Series of Potent and Selective TGF-β Type I Receptor Inhibitors

Françoise Gellibert, James M. Woolven, Marie-Hélène Fouchet et al. · Journal of Medicinal Chemistry · 2004 · 217 citations · Full text

Discovery and Lead-Optimization of 4,5-Dihydropyrazoles as Mono-Kinase Selective, Orally Bioavailable and Efficacious Inhibitors of Receptor Interacting Protein 1 (RIP1) Kinase

Philip A. Harris, Nicolas Faucher, Nicolas George et al. · Journal of Medicinal Chemistry · 2019 · 68 citations · Full text

Drug Target, Immunology, Efficacious Inhibitors +19

Discovery of novel indazole derivatives as dual angiotensin II antagonists and partial PPARγ agonists

Yann Lamotte, Nicolas Faucher, Julien Sançon et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 22 citations · Full text

Molecular Pharmacology, Novel Indazole Derivatives, Medicine +5

Discovery of Pyridones As Oral AMPK Direct Activators

Olivier Mirguet, Stéphane Sautet, Catherine-Anne Clément et al. · ACS Medicinal Chemistry Letters · 2013 · 14 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +11