Koppara Samuel

Extrapolation of Diclofenac Clearance from in Vitro Microsomal Metabolism Data: Role of Acyl Glucuronidation and Sequential Oxidative Metabolism of the Acyl Glucuronide

Sanjeev Kumar, Koppara Samuel, S. Ramaswamy et al. · Journal of Pharmacology and Experimental Therapeutics · 2002 · 165 citations

Discovery of <i>N</i>-[(1<i>S</i>,2<i>S</i>)-3-(4-Chlorophenyl)-2- (3-cyanophenyl)-1-methylpropyl]-2-methyl-2- {[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide (MK-0364), a Novel, Acyclic Cannabinoid-1 Receptor Inverse Agonist for the Treatment of Obesity

Linus S. Lin, Thomas J. Lanza, James P. Jewell et al. · Journal of Medicinal Chemistry · 2006 · 122 citations · Full text

Cannabis Use, Molecular Pharmacology, Medicinal Chemistry +15

Effects of dietary gallic acid supplementation on performance, antioxidant status, and jejunum intestinal morphology in broiler chicks

Koppara Samuel, J. Wang, Hui Yue et al. · Poultry Science · 2017 · 83 citations · Full text

Nutrition, Gastroenterology, Experimental Nutrition +19

Addressing the metabolic activation potential of new leads in drug discovery: a case study using ion trap mass spectrometry and tritium labeling techniques

Koppara Samuel, Wenji Yin, Ralph A. Stearns et al. · Journal of Mass Spectrometry · 2003 · 77 citations

Hit Identification, Metabolic Activation, Metabolomic Profiling +17

Hybrid-Designed Inhibitors of p38 MAP Kinase Utilizing<i>N</i>-Arylpyridazinones

Steven L. Colletti, Jessica L. Frie, Elizabeth C. Dixon et al. · Journal of Medicinal Chemistry · 2002 · 42 citations · Full text

Combinatorial Chemistry, Molecular Pharmacology, Medicinal Chemistry +15