Walaa R. Mahmoud

Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform

Hany S. Ibrahim, Heba Abdelrasheed Allam, Walaa R. Mahmoud et al. · European Journal of Medicinal Chemistry · 2018 · 69 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +11

Mechanistic selectivity investigation and 2D-QSAR study of some new antiproliferative pyrazoles and pyrazolopyridines as potential CDK2 inhibitors

Ghaneya S. Hassan, Hanan H. Georgey, Esraa Z. Mohammed et al. · European Journal of Medicinal Chemistry · 2021 · 50 citations · Full text

Medicinal Chemistry, Drug Target, 2D-qsar Study +11

Inhibition studies on a panel of human carbonic anhydrases with<i>N</i>1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails

Fadi M. Awadallah, Silvia Bua, Walaa R. Mahmoud et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 2018 · 48 citations · Full text

Design, synthesis, <i>in silico</i> docking, ADMET and anticancer evaluations of thiazolidine-2,4-diones bearing heterocyclic rings as dual VEGFR-2/EGFR^T790M tyrosine kinase inhibitors

Nada A. A. M. Aziz, Riham F. George, Khaled El‐Adl et al. · RSC Advances · 2022 · 42 citations · Full text

Synthesis and biological evaluation of some novel thiobenzimidazole derivatives as anti-renal cancer agents through inhibition of c-MET kinase

Hany S. Ibrahim, Mohamed E. Albakri, Walaa R. Mahmoud et al. · Bioorganic Chemistry · 2019 · 31 citations

Medicinal Chemistry, C-met Kinase, Novel Thiobenzimidazole Derivatives +10