Tiny J. P. Adolfs

Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel 3,4-Diarylpyrazolines as Potent and Selective CB₁ Cannabinoid Receptor Antagonists

Jos H.M. Lange, Hein K. A. C. Coolen, Herman H. van Stuivenberg et al. · Journal of Medicinal Chemistry · 2003 · 186 citations · Full text

Drug Target, Biological Properties, X-ray Diffraction Study +21

Bioisosteric Replacements of the Pyrazole Moiety of Rimonabant:  Synthesis, Biological Properties, and Molecular Modeling Investigations of Thiazoles, Triazoles, and Imidazoles as Potent and Selective CB₁Cannabinoid Receptor Antagonists

Jos H.M. Lange, Herman H. van Stuivenberg, Hein K. A. C. Coolen et al. · Journal of Medicinal Chemistry · 2004 · 177 citations · Full text

Pyrazole Series, Organic Chemistry, Pharmacotherapy +19

Novel 3,4-diarylpyrazolines as potent cannabinoid CB1 receptor antagonists with lower lipophilicity

Jos H.M. Lange, Herman H. van Stuivenberg, Willem Veerman et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 61 citations · Full text

Cannabis Use, Molecular Pharmacology, Medicinal Chemistry +12

7-Azaindole derivatives as potential partial nicotinic agonists

Axel R. Stoit, Arnold P. den Hartog, Harry Mons et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 17 citations · Full text

Molecular Pharmacology, Medicine, Nicotine +5