Vatee Pattaropong

Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines

Xiaohu Ouyang, Evgueni L. Piatnitski, Vatee Pattaropong et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 98 citations

Medicinal Chemistry, Polymer-drug Conjugate, Medicine +11

Discovery of AM-1638: A Potent and Orally Bioavailable GPR40/FFA1 Full Agonist

Sean P. Brown, Paul J. Dransfield, Marc Vimolratana et al. · ACS Medicinal Chemistry Letters · 2012 · 88 citations · Full text

Partial Agonist 1, Pancreatic Islets, Biochemistry +12

Discovery and in Vivo Evaluation of (<i>S</i>)-<i>N</i>-(1-(7-Fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9<i>H</i>-purin-6-amine (AMG319) and Related PI3Kδ Inhibitors for Inflammation and Autoimmune Disease

Timothy D. Cushing, Xiaolin Hao, Youngsook Shin et al. · Journal of Medicinal Chemistry · 2014 · 84 citations

Pharmaceutical Science, Immune Regulation, Immunology +23

Discovery and Optimization of Potent GPR40 Full Agonists Containing Tricyclic Spirocycles

Yingcai Wang, Jiwen Liu, Paul J. Dransfield et al. · ACS Medicinal Chemistry Letters · 2013 · 81 citations · Full text

Combinatorial Chemistry, Molecular Physiology, Biochemistry +13

Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors

Xiaohu Ouyang, Xiaoling Chen, Evgueni L. Piatnitski et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 69 citations

Medicinal Chemistry, Medicine, Natural Sciences +8