Andrea van de Stolpe

Catechol Pyrazolinones as Trypanocidals: Fragment-Based Design, Synthesis, and Pharmacological Evaluation of Nanomolar Inhibitors of Trypanosomal Phosphodiesterase B1

Kristina M. Orrling, Chimed Jansen, Xuan Lan Vu et al. · Journal of Medicinal Chemistry · 2012 · 56 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Molecular Determinants of Ligand Binding Modes in the Histamine H₄Receptor: Linking Ligand-Based Three-Dimensional Quantitative Structure–Activity Relationship (3D-QSAR) Models to in Silico Guided Receptor Mutagenesis Studies

Enade Perdana Istyastono, Saskia Nijmeijer, Herman D. Lim et al. · Journal of Medicinal Chemistry · 2011 · 52 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: Synthesis, pharmacological evaluation, and cross-target QSAR studies

Herman D. Lim, Enade Perdana Istyastono, Andrea van de Stolpe et al. · Bioorganic & Medicinal Chemistry · 2009 · 34 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Optical control of the β2-adrenergic receptor with opto-prop-2: A cis-active azobenzene analog of propranolol

Reggie Bosma, Nicola C. Dijon, Yang Zheng et al. · iScience · 2022 · 19 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Synthesis and pharmacological evaluation of some amino-acid-containing cyproheptadine derivatives as dual antagonists of histamine H1- and leukotriene D4-receptors

MQ Zhang, Andrea van de Stolpe, OP Zuiderveld et al. · European Journal of Medicinal Chemistry · 1997 · 16 citations

Medicine, Medicinal Chemistry, Pharmacology +12