Rebekah Carson

Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1

Lee D. Fader, Éric Malenfant, Mathieu Parisien et al. · ACS Medicinal Chemistry Letters · 2014 · 175 citations · Full text

Hiv-1 Integrase, Immunology, Molecular Biology +16

Compound Aggregation in Drug Discovery: Implementing a Practical NMR Assay for Medicinal Chemists

Steven R. LaPlante, Rebekah Carson, James Gillard et al. · Journal of Medicinal Chemistry · 2013 · 103 citations

Practical Nmr Assay, Pharmaceutical Science, Compound Aggregation +24

Monitoring Drug Self-Aggregation and Potential for Promiscuity in Off-Target In Vitro Pharmacology Screens by a Practical NMR Strategy

Steven R. LaPlante, Norman Aubry, Gordon T. Bolger et al. · Journal of Medicinal Chemistry · 2013 · 54 citations

Pharmaceutical Science, Pharmaceutical Research, Engineering +23

Palladium-Catalyzed Intramolecular Reactions of (<i>E</i>)-2,2-Disubstituted 1-Alkenyldimethylalanes with Aryl Triflates

Éric Fillion, V.E. Trepanier, Jarkko J. Heikkinen et al. · Organometallics · 2009 · 30 citations

Methyl Cross-coupling Reaction, Cross-coupling Reaction, Engineering +9

Aligning Potency and Pharmacokinetic Properties for Pyridine-Based NCINIs

Lee D. Fader, Murray D. Bailey, Eric Beaulieu et al. · ACS Medicinal Chemistry Letters · 2016 · 23 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Compound 2 +15