Hwang‐Fun Lu

Conformationally Constrained [<i>p</i>-(ω-Aminoalkyl)phenacetyl]-<scp>l</scp>-seryl-<scp>l</scp>-lysyl Dipeptide Amides as Potent Peptidomimetic Inhibitors of <i>Candida albicans</i> and Human Myristoyl-CoA:Protein <i>N</i>-Myristoyl Transferase

Srinivasan Nagarajan, Balekudru Devadas, Mark E. Zupec et al. · Journal of Medicinal Chemistry · 1997 · 44 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Synthesis and biological evaluation of substituted benzoxazoles as inhibitors of mPGES-1: Use of a conformation-based hypothesis to facilitate compound design

Daniel P. Walker, Graciela B. Arhancet, Hwang‐Fun Lu et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 27 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

R-Isomers of Arg-Gly-Asp (RGD) mimics as potent αvβ3 inhibitors

Srinivasan Nagarajan, Balekudru Devadas, James W. Malecha et al. · Bioorganic & Medicinal Chemistry · 2007 · 16 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective αvβ3 inhibitor: Design, synthesis, and optimization

Srinivasan Nagarajan, Hwang‐Fun Lu, Alan F. Gasiecki et al. · Bioorganic & Medicinal Chemistry · 2007 · 14 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Replacements for lysine in l-seryl-l-lysyl dipeptide amide inhibitors of candida albicans myristoyl-CoA:protein N-myristoyltransferase

David Brown, Balekudru Devadas, Hwang‐Fun Lu et al. · Bioorganic & Medicinal Chemistry Letters · 1997 · 12 citations

Pharmacy, Biochemistry, Medicinal Chemistry +10