Gustave Bergnes

Antitumor activity of an allosteric inhibitor of centromere-associated protein-E

Kenneth W. Wood, Latesh Lad, Lusong Luo et al. · Proceedings of the National Academy of Sciences · 2010 · 252 citations · Full text

Antitumor Activity, Cenp-e Motor Activity, Molecular Biology +18

Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295

Xiangping Qian, Andrew McDonald, Han-Jie Zhou et al. · ACS Medicinal Chemistry Letters · 2010 · 64 citations · Full text

Molecular Biology, New Generation, Cancer Biology +19

Creatine and phosphocreatine analogs: anticancer activity and enzymatic analysis.

Gustave Bergnes, Vrinda Khandekar, Margaret O'Keefe et al. · PubMed · 1996 · 30 citations

Substrate Analogs, Pharmacotherapy, Creatine Kinase +18

Generation of an Ugi library of phosphate mimic-containing compounds and identification of novel dual specific phosphatase inhibitors

Gustave Bergnes, Carla L. Gilliam, Michael D. Boisclair et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 29 citations

Medicinal Chemistry, Biosynthesis, Bioorganic Chemistry +12

Discovery of<i>Tirasemtiv</i>, the First Direct Fast Skeletal Muscle Troponin Activator

Scott E. Collibee, Gustave Bergnes, Alexander R. Muci et al. · ACS Medicinal Chemistry Letters · 2018 · 29 citations · Full text