Concepedia

Selective tumor targeting enabled by picomolar fibroblast activation protein inhibitors isolated from a DNA-encoded affinity maturation library

Sara Puglioli, Eleonore Schmidt, Christian Pellegrino, Luca Prati, Sebastian Oehler, Roberto De Luca, Andrea Galbiati, Claudia Comacchio, Lisa Nadal, Jörg Scheuermann,

Chem · 2022 · 41 citations · 38 references

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References

38

Lutetium-177–PSMA-617 for Metastatic Castration-Resistant Prostate Cancer

Oliver Sartor, Johann S. de Bono, Kim N. et al. · New England Journal of Medicine · 2021 · 2.6K citations · Full text

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Phase III Study of Docetaxel and Cisplatin Plus Fluorouracil Compared With Cisplatin and Fluorouracil As First-Line Therapy for Advanced Gastric Cancer: A Report of the V325 Study Group

Eric Van Cutsem, Vladimir Moiseyenko, Sergei Tjulandin et al. · Journal of Clinical Oncology · 2006 · 1.9K citations · Full text

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Encoded combinatorial chemistry.

Sydney Brenner, Richard A. Lerner · Proceedings of the National Academy of Sciences · 1992 · 1K citations

, , +17

Development of Quinoline-Based Theranostic Ligands for the Targeting of Fibroblast Activation Protein

Thomas Lindner, Anastasia Loktev, Annette Altmann et al. · Journal of Nuclear Medicine · 2018 · 920 citations · Full text

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ACE2 X-Ray Structures Reveal a Large Hinge-bending Motion Important for Inhibitor Binding and Catalysis

Paul Towler, Bart L. Staker, Sridhar G. Prasad et al. · Journal of Biological Chemistry · 2004 · 744 citations · Full text

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