Concepedia

Development of novel benzofuran-based SLC-0111 analogs as selective cancer-associated carbonic anhydrase isoform IX inhibitors

Moataz A. Shaldam, Wagdy M. Eldehna, Alessio Nocentini, Zainab M. Elsayed, Tamer M. Ibrahim, Rofaida Salem, Ramadan A. El-Domany, Clemente Capasso, Hatem A. Abdel‐Aziz, Claudiu T. Supuran

European Journal of Medicinal Chemistry · 2021 · 63 citations · 26 references

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References

26

Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays

Tim R. Mosmann · Journal of Immunological Methods · 1983 · 55.6K citations

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The Carbon Dioxide Hydration Activity of Carbonic Anhydrase

Raja G. Khalifah · Journal of Biological Chemistry · 1971 · 1.9K citations · Full text

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Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX

Jānis Leitāns, Andris Kazāks, Agnese Balode et al. · Journal of Medicinal Chemistry · 2015 · 201 citations

, , +16

Design, synthesis and anticancer evaluation of thieno[2,3-d]pyrimidine derivatives as dual EGFR/HER2 inhibitors and apoptosis inducers

Souad A. El‐Metwally, Khaled F. Saied, Ibrahim H. Eissa et al. · Bioorganic Chemistry · 2019 · 179 citations

, , +16

Novel coumarin-6-sulfonamides as apoptotic anti-proliferative agents: synthesis, <i>in vitro</i> biological evaluation, and QSAR studies

Ahmed Sabt, Omaima M. Abdelhafez, Radwan El‐Haggar et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 2018 · 110 citations · Full text

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