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Pharmacologic Characterization of JNJ-42226314, [1-(4-Fluorophenyl)indol-5-yl]-[3-[4-(thiazole-2-carbonyl)piperazin-1-yl]azetidin-1-yl]methanone, a Reversible, Selective, and Potent Monoacylglycerol Lipase Inhibitor

Ryan M. Wyatt, Ian Fraser, Natalie Welty, Brian Lord, Michelle Wennerholm, Steven W. Sutton, Michael K. Ameriks, Christine Dugovic, Sujin Yun, Allison White,

Journal of Pharmacology and Experimental Therapeutics · 2019 · 29 citations · 75 references

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References

75

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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A peripheral mononeuropathy in rat that produces disorders of pain sensation like those seen in man

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Characterization and localization of cannabinoid receptors in rat brain: a quantitative in vitro autoradiographic study

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Activity of norepinephrine-containing locus coeruleus neurons in behaving rats anticipates fluctuations in the sleep-waking cycle

Gary Aston‐Jones, F E Bloom · Journal of Neuroscience · 1981 · 2K citations · Full text

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