Bioorganic & Medicinal Chemistry Letters · 2019 · 55 citations · 29 references
PharmacyMedicinal ChemistryPharmacologyBioisosterismDrug DiscoveryStructure-activity RelationshipsAromatic BioisosteresBioisosteric DesignLead Compound DesignLigand-based DesignMolecular DockingTuberculosis PharmacotherapyBioisosteric Lead ModificationBioisosteric OptimizationMolecular Docking AnalysisPyrazine ChemistryPyrazole BioisosteresPyrazole ChemistryTriazole ChemistryTriazole Synthesis
29
A Diarylquinoline Drug Active on the ATP Synthase of <i>Mycobacterium tuberculosis</i>
Koen Andries, Peter Verhasselt, Jérôme Guillemont et al. · Science · 2004 · 2.2K citations · Full text