New efficient synthesis of 4-aminocarbonyl substituted 4H-3,1-benzoxazines by a Passerini 3CC/Staudinger/aza-Wittig sequence

The aza-Wittig reaction: an efficient tool for the construction of carbon–nitrogen double bonds

Francisco Palácios, Concepción Alonso, Domitila Aparicio et al. · Tetrahedron · 2006 · 386 citations

Natural Sciences, Chemistry, Medicinal Chemistry +15

Multicomponent reactions

Ilan Marek · Tetrahedron · 2005 · 249 citations

2-Amino-4<i>H</i>-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease

Sheryl J. Hays, Bradley W. Caprathe, John L. Gilmore et al. · Journal of Medicinal Chemistry · 1998 · 158 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +12

A versatile synthesis of fused triazolo derivatives by sequential Ugi/alkyne-azide cycloaddition reactions

Irini Akritopoulou‐Zanze, Vijaya Gracias, Stevan W. Djurić · Tetrahedron Letters · 2004 · 131 citations

Natural Sciences, Chemistry, Medicinal Chemistry +11

New Synthetic Technology for Efficient Construction of α-Hydroxy-β-amino Amides via the Passerini Reaction¹

J. Edward Semple, Timothy D. Owens, Khanh Hung Nguyen et al. · Organic Letters · 2000 · 116 citations

Life Sciences, Biochemistry, Medicinal Chemistry +12