Concepedia

Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38α and BRD4

Stephanie M. Myers, Duncan C. Miller, Lauren Molyneux, Mercedes Arasta, Ruth H. Bawn, Timothy J. Blackburn, Simon J. Cook, Noel Edwards, Jane Endicott, Bernard T. Golding,

European Journal of Medicinal Chemistry · 2019 · 21 citations · 32 references

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32

<i>XDS</i>

Wolfgang Kabsch · Acta Crystallographica Section D Biological Crystallography · 2010 · 16.5K citations · Full text

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Overview of the<i>CCP</i>4 suite and current developments

Martyn Winn, Charles Ballard, Kevin Cowtan et al. · Acta Crystallographica Section D Biological Crystallography · 2011 · 12.4K citations · Full text

The Cambridge Structural Database

Colin R. Groom, Ian Bruno, Matthew P. Lightfoot et al. · Acta Crystallographica Section B Structural Science Crystal Engineering and Materials · 2016 · 9.8K citations · Full text

Molecular replacement with<i>MOLREP</i>

Alexei A. Vagin, A. Teplyakov · Acta Crystallographica Section D Biological Crystallography · 2009 · 3.6K citations

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Data processing and analysis with the<i>autoPROC</i>toolbox

Clemens Vonrhein, Claus Flensburg, Peter M. Keller et al. · Acta Crystallographica Section D Biological Crystallography · 2011 · 2K citations · Full text

, , +21