Concepedia

N-Acyl pyrazoles: Effective and tunable inhibitors of serine hydrolases

Katerina Otrubova, Shreyosree Chatterjee, Srijana Ghimire, Benjamin F. Cravatt, Dale L. Boger

Bioorganic & Medicinal Chemistry · 2019 · 26 citations · 75 references

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References

75

Isolation and Structure of a Brain Constituent That Binds to the Cannabinoid Receptor

William A. Devane, Aviva Breuer, Roger G. Pertwee et al. · Science · 1992 · 5.6K citations

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Identification of an endogenous 2-monoglyceride, present in canine gut, that binds to cannabinoid receptors

Raphael Mechoulam, Shimon Ben‐Shabat, L Hanŭs et al. · Biochemical Pharmacology · 1995 · 2.9K citations

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2-Arachidonoylgylcerol: A Possible Endogenous Cannabinoid Receptor Ligand in Brain

Takayuki Sugiura, Shigeru Kondo, Akihiro Sukagawa et al. · Biochemical and Biophysical Research Communications · 1995 · 2.2K citations

, , +9

Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides

Benjamin F. Cravatt, Dan K. Giang, Stephen P. Mayfield et al. · Nature · 1996 · 2.1K citations

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A Comprehensive Profile of Brain Enzymes that Hydrolyze the Endocannabinoid 2-Arachidonoylglycerol

Jacqueline L. Blankman, Gabriel M. Simon, Benjamin F. Cravatt · Chemistry & Biology · 2007 · 1.2K citations · Full text

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