European Journal of Medicinal Chemistry · 2018 · 24 citations · 27 references
PharmacyMedicinal ChemistryPharmacologyDrug DiscoveryMolecular PharmacologyStructure-activity RelationshipsEnzyme InhibitionHit-to-lead OptimizationLead Compound DesignLead DiscoveryPotency OptimizationStereochemical OptimizationChemical Synthesis Of AnaloguesEnzyme Inhibitor DiscoveryHit-to-lead Library ExpansionMedicinal Chemistry ApplicationsTyrosine-targeted Inhibitors
27
PTP1B Regulates Leptin Signal Transduction In Vivo
Janice M. Zabolotny, Kendra K. Bence, Alain Stricker‐Krongrad et al. · Developmental Cell · 2002 · 820 citations · Full text
Discovery of a Small Molecule Insulin Mimetic with Antidiabetic Activity in Mice
Bei Zhang, Gino Salituro, Deborah Szalkowski et al. · Science · 1999 · 455 citations