Concepedia

Discovery of novel arylethenesulfonyl fluorides as potential candidates against methicillin-resistant of Staphylococcus aureus (MRSA) for overcoming multidrug resistance of bacterial infections

Gao‐Feng Zha, Shi‐Meng Wang, K.P. Rakesh, Syed Nasir Abbas Bukhari, H.M. Manukumar, N. Mallesha, Hua‐Li Qin

European Journal of Medicinal Chemistry · 2018 · 91 citations · 33 references

DOI

Concepts

References

33

The Epidemic of Antibiotic-Resistant Infections: A Call to Action for the Medical Community from the Infectious Diseases Society of America

Brad Spellberg, R. Guidos, David N. Gilbert et al. · Clinical Infectious Diseases · 2007 · 1.6K citations · Full text

, , +21

PHASE: a new engine for pharmacophore perception, 3D QSAR model development, and 3D database screening: 1. Methodology and preliminary results

Steven L. Dixon, Alexander M. Smondyrev, Eric H. Knoll et al. · Journal of Computer-Aided Molecular Design · 2006 · 1.2K citations

, , +11

Sulfonyl fluorides as privileged warheads in chemical biology

Arjun Narayanan, Lyn H. Jones · Chemical Science · 2015 · 524 citations · Full text

Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes

Qian Zhao, Xiaohu Ouyang, Xiaobo Wan et al. · Journal of the American Chemical Society · 2017 · 358 citations

, , +21

“Inverse Drug Discovery” Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates

D.E. Mortenson, Gabriel J. Brighty, Lars Plate et al. · Journal of the American Chemical Society · 2017 · 299 citations · Full text