Concepedia

Evaluation of Carbazeran 4-Oxidation and O6-Benzylguanine 8-Oxidation as Catalytic Markers of Human Aldehyde Oxidase: Impact of Cytosolic Contamination of Liver Microsomes

Jiarong Xie, Nur Fazilah Saburulla, Shiyan Chen, Siew Ying Wong, Ze Ping Yap, Linghua Harris Zhang, Aik Jiang Lau

Drug Metabolism and Disposition · 2018 · 26 citations · 38 references

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References

38

Steroid hormone hydroxylase specificities of eleven cDNA-expressed human cytochrome P450s

David J. Waxman, D P Lapenson, Toshifumi Aoyama et al. · Archives of Biochemistry and Biophysics · 1991 · 324 citations

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Effect of common organic solvents on in vitro cytochrome P450-mediated metabolic activities in human liver microsomes.

Nathalie Chauret, Annick Gauthier, Deborah A. Nicoll‐Griffith · PubMed · 1998 · 310 citations

, , +16

Nonspecific binding to microsomes: impact on scale-up of in vitro intrinsic clearance to hepatic clearance as assessed through examination of warfarin, imipramine, and propranolol.

R S Obach · PubMed · 1997 · 281 citations

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Furafylline is a potent and selective inhibitor of cytochrome P450IA2 in man.

Dorothea Sesardic, B. P. Murray, Sandra Murray et al. · British Journal of Clinical Pharmacology · 1990 · 280 citations · Full text

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Isoform-selective mechanism-based inhibition of human cytochrome P450 1A2 by furafylline

Kent L. Kunze, William Trager · Chemical Research in Toxicology · 1993 · 220 citations

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