Concepedia

Structure-based design and profiling of novel 17β-HSD14 inhibitors

Florian Braun, Nicole Bertoletti, Gabriele Möller, Jerzy Adamski, Martin Frotscher, Nathalie Guragossian, Patrícia Alexandra Madeira Gírio, Marc Le Borgne, Laurent Ettouati, Pierre Falson,

European Journal of Medicinal Chemistry · 2018 · 14 citations · 32 references

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32

Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays

Tim R. Mosmann · Journal of Immunological Methods · 1983 · 55.6K citations

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Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Molecular Properties That Influence the Oral Bioavailability of Drug Candidates

Daniel F. Veber, Stephen R. Johnson, Hung‐Yuan Cheng et al. · Journal of Medicinal Chemistry · 2002 · 8.1K citations

, , +15

UniProt: the Universal Protein knowledgebase

Rolf Apweiler · Nucleic Acids Research · 2003 · 7.8K citations · Full text

, , +11

UniProt: the universal protein knowledgebase

Nucleic Acids Research · 2016 · 4.7K citations · Full text

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