Concepedia

Discovery of novel anti-tuberculosis agents with pyrrolo[1,2-a]quinoxaline-based scaffold

Ting Wang, Yunxiang Tang, Yang Yang, Qi An, Zitai Sang, Tao Yang, Pingxian Liu, Tianyu Zhang, Yong Deng, Youfu Luo

Bioorganic & Medicinal Chemistry Letters · 2018 · 52 citations · 17 references

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References

17

High throughput artificial membrane permeability assay for blood–brain barrier

Li Di, Edward H. Kerns, Kristi Fan et al. · European Journal of Medicinal Chemistry · 2003 · 1.1K citations

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Multidrug-resistant and extensively drug-resistant tuberculosis: a threat to global control of tuberculosis

Neel R. Gandhi, Paul Nunn, Keertan Dheda et al. · The Lancet · 2010 · 1K citations

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Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis

Kévin Pethe, Pablo Bifani, Jichan Jang et al. · Nature Medicine · 2013 · 595 citations · Full text

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Computational methods for the prediction of ‘drug-likeness’

David E. Clark, Stephen D. Pickett · Drug Discovery Today · 2000 · 569 citations

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Comparison of blood–brain barrier permeability assays: in situ brain perfusion, MDR1-MDCKII and PAMPA-BBB

Li Di, Edward H. Kerns, Ian F. Bezar et al. · Journal of Pharmaceutical Sciences · 2008 · 153 citations

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