Concepedia

The opioid receptor triple agonist DPI-125 produces analgesia with less respiratory depression and reduced abuse liability

Shou-Pu Yi, Qinghong Kong, Yulei Li, Chenling Pan, Jie Yu, Benqiang Cui, Yingfei Wang, Guanlin Wang, Peilan Zhou, Lili Wang,

Acta Pharmacologica Sinica · 2017 · 15 citations · 50 references

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Concepts

References

50

A Rapid and Sensitive Method for the Quantitation of Microgram Quantities of Protein Utilizing the Principle of Protein-Dye Binding

Mark A. Bradford · Analytical Biochemistry · 1976 · 225.4K citations

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

Marion M. Bradford · Analytical Biochemistry · 1976 · 211.2K citations

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Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Crystal structure of the µ-opioid receptor bound to a morphinan antagonist

Aashish Manglik, Andrew C. Kruse, Tong Sun Kobilka et al. · Nature · 2012 · 1.4K citations

, , +14

Structural insights into µ-opioid receptor activation

Weijiao Huang, Aashish Manglik, AJ Venkatakrishnan et al. · Nature · 2015 · 911 citations · Full text

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