Concepedia

A new series of pyridinyl-alkynes as antagonists of the metabotropic glutamate receptor 5 (mGluR5)

Peter Bach, Karolina Nilsson, Andreas Wållberg, Udo Bauer, Lance G. Hammerland, Alecia Peterson, Tor Svensson, Krister Österlund, David Karis, Maria Boije,

Bioorganic & Medicinal Chemistry Letters · 2006 · 31 citations · 20 references

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20

A convenient synthesis of acetylenes: catalytic substitutions of acetylenic hydrogen with bromoalkenes, iodoarenes and bromopyridines

Kenkichi Sonogashira, Yasuo Tohda, Nobue Hagihara · Tetrahedron Letters · 1975 · 5.1K citations

, , +11

A family of metabotropic glutamate receptors

Yasuto Tanabe, Masayuki Masu, Takahiro Ishii et al. · Neuron · 1992 · 929 citations

, , +12

A family of metabotropic glutamate receptors

康人 田辺 · Medical Entomology and Zoology · 1992 · 879 citations

, , +12

Molecular characterization of a novel metabotropic glutamate receptor mGluR5 coupled to inositol phosphate/Ca2+ signal transduction.

Takaaki Abe, Hidemitsu Sugihara, Hiroyuki Nawa et al. · Journal of Biological Chemistry · 1992 · 811 citations · Full text

, , +17

2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist

F. Gasparini, Kurt Lingenhöhl, Natacha Stoehr et al. · Neuropharmacology · 1999 · 720 citations

, , +7