Krister Österlund

Asymmetric Total Synthesis of (+)-Tolterodine, a New Muscarinic Receptor Antagonist, via Copper-Assisted Asymmetric Conjugate Addition of Aryl Grignard Reagents to 3-Phenyl-prop-2-enoyl-oxazolidinones

Pher G. Andersson, Hans E. Schink, Krister Österlund · The Journal of Organic Chemistry · 1998 · 75 citations

Molecular Pharmacology, Medicinal Chemistry, Asymmetric Total Synthesis +13

Lead Optimization of Ethyl 6-Aminonicotinate Acyl Sulfonamides as Antagonists of the P2Y₁₂ Receptor. Separation of the Antithrombotic Effect and Bleeding for Candidate Drug AZD1283

Peter Bach, Thomas Antonsson, Ruth Bylund et al. · Journal of Medicinal Chemistry · 2013 · 63 citations · Full text

Pharmaceutical Science, Pharmacotherapy, Pharmaceutical Chemistry +20

A new series of pyridinyl-alkynes as antagonists of the metabotropic glutamate receptor 5 (mGluR5)

Peter Bach, Karolina Nilsson, Andreas Wållberg et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 31 citations · Full text

Biochemistry, Functional Selectivity, Medicine +9

Identification of pyrazolo-pyrimidinones as GHS-R1a antagonists and inverse agonists for the treatment of obesity

William McCoull, Peter Barton, Anders Broo et al. · MedChemComm · 2012 · 25 citations

Inverse Agonists, Immunology, Food Intake +20

Structure–activity relationships for the linker in a series of pyridinyl-alkynes that are antagonists of the metabotropic glutamate receptor 5 (mGluR5)

Peter Bach, Karolina Nilsson, Tor Svensson et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 22 citations · Full text

Molecular Pharmacology, Biochemistry, Medicine +11