Concepedia
European Journal of Medicinal Chemistry · 2005 · 101 citations · 8 references
PharmacyMedicinal ChemistryPharmacologyBioisosterismOrganic ChemistrySynthetic Medicinal ChemistryAromatic BioisosteresBioisosteric DesignClassical BioisosteresAntiprotozoal ChemotherapyAntiprotozoal PharmacologyBenzimidazole ChemistryBenzimidazole Synthesis
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Synthesis and antiparasitic activity of 2-(Trifluoromethyl)benzimidazole derivatives
Gabriel Navarrete‐Vázquez, Roberto Cedillo, Alicia Hernández‐Campos et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 206 citations
Pharmacy, Chemistry, Medicinal Chemistry +12
In vitro activities of and mechanisms of resistance to antifol antimalarial drugs
Wilbur K. Milhous, Norman F. Weatherly, Jean H. Bowdre et al. · Antimicrobial Agents and Chemotherapy · 1985 · 197 citations
Life Sciences, Biochemistry, Pharmacology +14
Plasmodium falciparum: Induction of resistance to mefloquine in cloned strains by continuous drug exposure in vitro
A.M.J. Oduola, Wilbur K. Milhous, Norman F. Weatherly et al. · Experimental Parasitology · 1988 · 143 citations
Medicine, Infectious Diseases, Pharmacology +16
Synthesis, antiprotozoal and anticancer activity of substituted 2-trifluoromethyl- and 2-pentafluoroethylbenzimidazoles
Mariola Andrzejewska · European Journal of Medicinal Chemistry · 2002 · 132 citations
Pharmacy, Medicinal Chemistry, Pharmacology +11
Synthesis, antiprotozoal and antibacterial activity of nitro- and halogeno-substituted benzimidazole derivatives.
Zygmunt Kazimierczuk, Jacqueline Upcroft, Peter Upcroft et al. · Acta Biochimica Polonica · 2002 · 118 citations · Full text
Medicine, Microbiology, Pharmacology +10