Concepedia

Synthesis and SAR of highly potent and selective dopamine D3-receptor antagonists: 1H-Pyrimidin-2-one derivatives

Hervé Geneste, Gisela Backfisch, Wilfried M. Braje, Jürgen Delzer, Andreas Haupt, Charles W. Hutchins, Linda L. King, Andreas Kling, H. J. Teschendorf, Liliane Unger,

Bioorganic & Medicinal Chemistry Letters · 2005 · 17 citations · 12 references

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12

Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties

Peter Ertl, Bernhard Rohde, Paul M. Selzer · Journal of Medicinal Chemistry · 2000 · 3K citations

, , +19

Caco-2 Cell Monolayers as a Model for Drug Transport Across the Intestinal Mucosa

Allen R. Hilgers, Robert A. Conradi, Philip S. Burton · Pharmaceutical Research · 1990 · 579 citations

Pharmacological Actions of a Novel, High-Affinity, and Selective Human Dopamine D3 Receptor Antagonist, SB-277011-A

C. Reavill, Stephen G. Taylor, Martyn Wood et al. · Journal of Pharmacology and Experimental Therapeutics · 2000 · 288 citations · Full text

<i>N</i>-(ω-(4-(2-Methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as Dopamine D<sub>2</sub> and D<sub>3</sub> Receptor Ligands

Anneke E. Hackling, Robin Ghosh, Sylvie Perachon et al. · Journal of Medicinal Chemistry · 2003 · 103 citations · Full text

The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors

Karsten Wicke, J. Garcia-Ladona · European Journal of Pharmacology · 2001 · 74 citations

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