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Discovery, synthesis and SAR of azinyl- and azolylbenzamides antagonists of the P2X7 receptor

Chakrapani Subramanyam, Allen J. Duplantier, Mark A. Dombroski, Shang-Poa Chang, Christopher A. Gabel, Carrie Whitney‐Pickett, David G. Perregaux, Jeff M. Labasi, Kwansik Yoon, Richard M. Shepard,

Bioorganic & Medicinal Chemistry Letters · 2011 · 20 citations · 12 references

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12

Molecular Properties That Influence the Oral Bioavailability of Drug Candidates

Daniel F. Veber, Stephen R. Johnson, Hung‐Yuan Cheng et al. · Journal of Medicinal Chemistry · 2002 · 8.1K citations

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Receptors for Purines and Pyrimidines

Geoffrey Burnstock, Alexei Verkhratsky · 2012 · 4K citations

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Palladium(0)-Catalyzed Cross-Coupling Reaction of Alkoxydiboron with Haloarenes: A Direct Procedure for Arylboronic Esters

Tatsuo Ishiyama, Miki Murata, Norio Miyaura · The Journal of Organic Chemistry · 1995 · 1.6K citations

, , +14

Altered Cytokine Production in Mice Lacking P2X7Receptors

Mike Solle, Jeff M. Labasi, David G. Perregaux et al. · Journal of Biological Chemistry · 2001 · 925 citations · Full text

, , +17

Prediction of Volume of Distribution Values in Humans for Neutral and Basic Drugs Using Physicochemical Measurements and Plasma Protein Binding Data

Franco Lombardo, R. Scott Obach, Marina Shalaeva et al. · Journal of Medicinal Chemistry · 2002 · 209 citations

, , +17