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Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist

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Operational models of pharmacological agonism

J.W. Black, P. Leff · Proceedings of the Royal Society of London. Series B, Biological sciences · 1983 · 1.1K citations

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Aripiprazole, a Novel Antipsychotic, Is a High-Affinity Partial Agonist at Human Dopamine D2 Receptors

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Ligand-specific regulation of the extracellular surface of a G-protein-coupled receptor

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