Concepedia

Activation of 9-[(R)-2-[[(S)-[[(S)-1-(Isopropoxycarbonyl)ethyl]amino] phenoxyphosphinyl]-methoxy]propyl]adenine (GS-7340) and Other Tenofovir Phosphonoamidate Prodrugs by Human Proteases

Gabriel Birkuš, Nilima Kutty, Gong-Xin He, Andrew Mulato, William Lee, Martin J. McDermott, Tomáš Cihlář

Molecular Pharmacology · 2008 · 99 citations · 30 references

DOI

Concepts

References

30

On the size of the active site in proteases. I. Papain

Israël Schechter, Arieh Berger · Biochemical and Biophysical Research Communications · 1967 · 5.2K citations

, , +9

Granules of the Human Neutrophilic Polymorphonuclear Leukocyte

Niels Borregaard, Jack B. Cowland · Blood · 1997 · 1.5K citations · Full text

, , +9

Biochemistry of dystrophic muscle. Mitochondrial succinate-tetrazolium reductase and adenosine triphosphatase

RJ Pennington · Biochemical Journal · 1961 · 1K citations · Full text

, , +17

L-<i>trans</i>-Epoxysuccinyl-leucylamido(4-guanidino)butane (E-64) and its analogues as inhibitors of cysteine proteinases including cathepsins B, H and L

A. John Barrett, A A Kembhavi, M A Brown et al. · Biochemical Journal · 1982 · 1K citations · Full text

, , +17

Structural and functional aspects of papain-like cysteine proteinases and their protein inhibitors.

Boris Turk, V Turk · PubMed · 1997 · 441 citations

, , +16