Concepedia
Drug Metabolism and Disposition · 2014 · 19 citations · 27 references
Open access
27
Human cytochrome P450 CYP2A13: predominant expression in the respiratory tract and its high efficiency metabolic activation of a tobacco-specific carcinogen, 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone.
Ta‐Chen Su, Ziping Bao, Qingyu Zhang et al. · PubMed · 2000 · 342 citations
Nasal Mucosa, Toxicological Mechanism, Respiratory Toxicology +16
Preclinical experimental models of drug metabolism and disposition in drug discovery and development
Donglu Zhang, Gang Luo, Xinxin Ding et al. · Acta Pharmaceutica Sinica B · 2012 · 292 citations · Full text
Medicinal Chemistry, Drug Target, Pharmacokinetic Modeling +15
Efficient activation of aflatoxin B<sub>1</sub> by cytochrome P450 2A13, an enzyme predominantly expressed in human respiratory tract
Xiaoyang He, Lili Tang, Shoulin Wang et al. · International Journal of Cancer · 2005 · 132 citations · Full text
Immunochemical characterization of multiple forms of cytochrome P-450 in rabbit nasal microsomes and evidence for tissue-specific expression of P-450s NMa and NMb.
Xinxin Ding, Minor J. Coon · Molecular Pharmacology · 1990 · 107 citations
Determination of the Role of Target Tissue Metabolism in Lung Carcinogenesis Using Conditional Cytochrome <i>P</i> 450 Reductase-Null Mice
Yan Weng, Cheng Fang, Robert J. Turesky et al. · Cancer Research · 2007 · 94 citations