Concepedia

Imetit and N-methyl derivatives. The transition from potent agonist to antagonist at histamine H3 receptors.1

C. Robin Ganellin, Benny Bang‐Andersen, Y. S. KHALAF, W. Tertiuk, J.M. Arrang, M. Garbarg, Xavier Ligneau, A. Rouleau, J.C. Schwartz

Bioorganic & Medicinal Chemistry Letters · 1992 · 22 citations · 9 references

DOI

Concepts

References

9

Definition and Antagonism of Histamine H2-receptors

J. W. Black, W. A. M. Duncan, C. J. DURANT et al. · Nature · 1972 · 2.3K citations

, , +12

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

, , +14

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 902 citations

, , +15

RECEPTORS MEDIATING SOME ACTIONS OF HISTAMINE

A. S. F. Ash, H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1966 · 766 citations · Full text

, , +12

Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists

Rodney C. Young, Robert Cameron Mitchell, Thomas H. Brown et al. · Journal of Medicinal Chemistry · 1988 · 522 citations

, , +15