Concepedia

HIGHLY SELECTIVE INHIBITION OF HUMAN CYP3A IN VITRO BY AZAMULIN AND EVIDENCE THAT INHIBITION IS IRREVERSIBLE

David M. Stresser, Marc I. Broudy, Thuy Ho, Catherine E. Cargill, Andrew P. Blanchard, Raman Sharma, Andre Dandeneau, Joseph Goodwin, Stephanie D. Turner, John C. L. Erve,

Drug Metabolism and Disposition · 2004 · 128 citations · 32 references

DOI

Concepts

References

32

THE CONDUCT OF IN VITRO AND IN VIVO DRUG-DRUG INTERACTION STUDIES: A PHARMACEUTICAL RESEARCH AND MANUFACTURERS OF AMERICA (PhRMA) PERSPECTIVE

Thorir D. Bjornsson, John T. Callaghan, Heidi J. Einolf et al. · Drug Metabolism and Disposition · 2003 · 784 citations

, , +17

Cytochrome P450 inhibitors. Evaluation of specificities in the in vitrometabolism of therapeutic agents by human liver microsomes.

Deborah J. Newton, R W Wang, Anthony Y.H. Lu · Drug Metabolism and Disposition · 1995 · 606 citations

, , +17

Microtiter Plate Assays for Inhibition of Human, Drug-Metabolizing Cytochromes P450

Charles L. Crespi, Vaughn P. Miller, Bruce W. Penman · Analytical Biochemistry · 1997 · 408 citations

, , +12

[10] Mechanism-based enzyme inactivators

Richard B. Silverman · Methods in enzymology on CD-ROM/Methods in enzymology · 1995 · 383 citations

, , +10

Cytochrome P450 isoform inhibitors as a tool for the investigation of metabolic reactions catalyzed by human liver microsomes.

Martine Bourrié, Viviane Meunier, Yves Berger et al. · Journal of Pharmacology and Experimental Therapeutics · 1996 · 362 citations

, , +15