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Influenza Neuraminidase Inhibitors Possessing a Novel Hydrophobic Interaction in the Enzyme Active Site:  Design, Synthesis, and Structural Analysis of Carbocyclic Sialic Acid Analogues with Potent Anti-Influenza Activity

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Anti-Influenza Prodrug Oseltamivir Is Activated by Carboxylesterase Human Carboxylesterase 1, and the Activation Is Inhibited by Antiplatelet Agent Clopidogrel

Deshi Shi, Jian Yang, Dongfang Yang et al. · Journal of Pharmacology and Experimental Therapeutics · 2006 · 277 citations · Full text

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Identification of GS 4104 as an Orally Bioavailable Prodrug of the Influenza Virus Neuraminidase Inhibitor GS 4071

Weixing Li, Paul A. Escarpe, Eugene Eisenberg et al. · Antimicrobial Agents and Chemotherapy · 1998 · 224 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +14

Development of a New Radioligand, <i>N</i>-(5-Fluoro-2-phenoxyphenyl)-<i>N</i>-(2-[¹⁸F]fluoroethyl-5-methoxybenzyl)acetamide, for PET Imaging of Peripheral Benzodiazepine Receptor in Primate Brain

Ming‐Rong Zhang, Jun Maeda, Masanao Ogawa et al. · Journal of Medicinal Chemistry · 2004 · 145 citations · Full text

Medicine, Neuroscience, Pharmacology +9

[11C]DAA1106: radiosynthesis and in vivo binding to peripheral benzodiazepine receptors in mouse brain

Ming‐Rong Zhang, Takayo Kida, Junko Noguchi et al. · Nuclear Medicine and Biology · 2003 · 142 citations · Full text

Medicine, Neuroscience, Pharmacology +10