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Identification of SD-0006, a potent diaryl pyrazole inhibitor of p38 MAP kinase

John K. Walker, Shaun R. Selness, Rajesh Devraj, Michael Hepperle, Win Naing, H.-S. Shieh, Ravi Kurambail, Syaulan Yang, Daniel L. Flynn, Alan G. Benson,

Bioorganic & Medicinal Chemistry Letters · 2010 · 21 citations · 8 references

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8

Differential Expression and Activation of p38 Mitogen-Activated Protein Kinase α, β, γ, and δ in Inflammatory Cell Lineages

Karin K. Hale, David Trollinger, Marynette Rihanek et al. · The Journal of Immunology · 1999 · 246 citations · Full text

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Pyrimidinylimidazole inhibitors of CSBP/P38 kinase demonstrating decreased inhibition of hepatic cytochrome P450 enzymes

Jerry L. Adams, Jeffrey C. Boehm, Shouki Kassis et al. · Bioorganic & Medicinal Chemistry Letters · 1998 · 113 citations · Full text

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Chemical Genetics Define the Roles of p38α and p38β in Acute and Chronic Inflammation

Stephen J. O’Keefe, John S. Mudgett, Susan Cupo et al. · Journal of Biological Chemistry · 2007 · 80 citations · Full text

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Effects of RWJ 67657, a p38 mitogen activated protein kinase (MAPK) inhibitor, on the production of inflammatory mediators by rheumatoid synovial fibroblasts

Johanna Westra · Annals of the Rheumatic Diseases · 2004 · 66 citations · Full text

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Synthesis, Crystal Structure, and Activity of Pyrazole-Based Inhibitors of p38 Kinase

Matthew J. Graneto, Ravi G. Kurumbail, Michael L. Vazquez et al. · Journal of Medicinal Chemistry · 2007 · 64 citations · Full text

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