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Synthesis and biological activity of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 2: 2′-Substituted triclosan derivatives

Joel S. Freundlich, Min Yu, Edinson Lucumi, Mack Kuo, Han-Chun Tsai, Juan‐Carlos Valderramos, Luchezar Karagyozov, William R. Jacobs, Guy A. Schiehser, David A. Fidock,

Bioorganic & Medicinal Chemistry Letters · 2006 · 54 citations · 15 references

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15

Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures<sup>1</sup>

Ahmed F. Abdel‐Magid, Kenneth G. Carson, Bruce D. Harris et al. · The Journal of Organic Chemistry · 1996 · 1.5K citations

, , +10

Triclosan offers protection against blood stages of malaria by inhibiting enoyl-ACP reductase of Plasmodium falciparum

Namita Surolia, Avadhesha Surolia · Nature Medicine · 2001 · 403 citations

, , +14

Targeting Tuberculosis and Malaria through Inhibition of Enoyl Reductase

Mack Kuo, Héctor R. Morbidoni, David Alland et al. · Journal of Biological Chemistry · 2003 · 262 citations · Full text

, , +15

Structural Elucidation of the Specificity of the Antibacterial Agent Triclosan for Malarial Enoyl Acyl Carrier Protein Reductase

Remo Perozzo, Mack Kuo, Amar Bir Singh Sidhu et al. · Journal of Biological Chemistry · 2002 · 212 citations · Full text

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TRICLOSAN AS A SUBSTRATE AND INHIBITOR OF 3′-PHOSPHOADENOSINE 5′-PHOSPHOSULFATE-SULFOTRANSFERASE AND UDP-GLUCURONOSYL TRANSFERASE IN HUMAN LIVER FRACTIONS

Liquan Wang, Charles N. Falany, Margaret O. James · Drug Metabolism and Disposition · 2004 · 188 citations

, , +13