Synthesis of new bridged tetrahydro-β-carbolines and spiro -fused quinuclidines

Rapid chromatographic technique for preparative separations with moderate resolution

W. Clark Still, Michaël Kahn, Abhijit Mitra · The Journal of Organic Chemistry · 1978 · 5.8K citations

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Synthesis and biological activity of 1,2,4-oxadiazole derivatives: highly potent and efficacious agonists for cortical muscarinic receptors

R. BAKER, T. BOOK, Clare O. Kneen et al. · Journal of Medicinal Chemistry · 1990 · 133 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Potent, Selective Tetrahydro-β-carboline Antagonists of the Serotonin 2B (5HT_2B) Contractile Receptor in the Rat Stomach Fundus

James E. Audia, Deborah A. Evrard, Gwyn R. Murdoch et al. · Journal of Medicinal Chemistry · 1996 · 119 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

A Rapid Total Synthesis of Spirotryprostatin B: Proof of Its Relative and Absolute Stereochemistry

Franz von Nussbaum, Samuel J. Danishefsky · Angewandte Chemie International Edition · 2000 · 117 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8

Three-dimensional quantitative structure-activity relationships of 5-HT receptor binding data for tetrahydropyridinylindole derivatives: a comparison of the Hansch and CoMFA methods

Atul Agarwal, Philip P. Pearson, Ethan Will Taylor et al. · Journal of Medicinal Chemistry · 1993 · 71 citations · Full text

Medicine, Chemistry, Pharmacology +13