Concepedia

Ligand Efficacy and Potency at Recombinant α2 Adrenergic Receptors

Jeffrey R. Jasper, John Lesnick, Leon Chang, Susan S Yamanishi, Thomas K. H. Chang, Sherry Hsu, David A. Daunt, Douglas W. Bonhaus, Richard M. Eglen

Biochemical Pharmacology · 1998 · 156 citations · 28 references

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References

28

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Type-Specific Regulation of Adenylyl Cyclase by G Protein βγ Subunits

Wei‐Jen Tang, Alfred G. Gilman · Science · 1991 · 1.1K citations

, , +15

Forskolin: its biological and chemical properties.

Seamon Kb, Daly Jw · PubMed · 1986 · 571 citations

, , +2

Modulation by mu-opioid agonists of guanosine-5'-O-(3-[35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells.

John R. Traynor, Stefan R. Nahorski · Molecular Pharmacology · 1995 · 462 citations

, , +17

Cloning and expression of a human kidney cDNA for an alpha 2-adrenergic receptor subtype.

John W. Regan, Tong Sun Kobilka, T L Yang-Feng et al. · Proceedings of the National Academy of Sciences · 1988 · 436 citations · Full text

, , +13