Asymmetric synthesis of α-hydroxy- phosphonamides, phosphonates and phosphonic acids

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

Bernd Stowasser, Karl‐Heinz Budt, Jianqi Li et al. · Tetrahedron Letters · 1992 · 407 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +13

Preparation of peptidic α-hydroxy phosphonates a new class of transition state analog renin inhibitors

Dinesh V. Patel, Katherine Rielly-Gauvin, Denis E. Ryono · Tetrahedron Letters · 1990 · 237 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

OPTICALLY ACTIVE 1-AMINOALKYLPHOSPHONIC ACIDS

Balram Dhawan, Derek Redmore · Phosphorous and Sulfur and the Related Elements · 1987 · 178 citations

Life Sciences, Biochemistry, Pharmacology +15

Design and reactivity of topologically unique, chiral phosphonamides. Remarkable diastereofacial selectivity in asymmetric olefination and alkylation

Stephen Hanessian, Daniel Delorme, Serge Beaudoin et al. · Journal of the American Chemical Society · 1984 · 163 citations

Pharmacy, Chemistry, Medicinal Chemistry +7

Phosphonopeptides as Antibacterial Agents: Mechanism of Action of Alaphosphin

F. R. Atherton, Michael J. Hall, Cedric H. Hassall et al. · Antimicrobial Agents and Chemotherapy · 1979 · 153 citations · Full text

Life Sciences, Microbiology, Pharmacology +15