Karl‐Heinz Budt

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

Bernd Stowasser, Karl‐Heinz Budt, Jianqi Li et al. · Tetrahedron Letters · 1992 · 407 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +13

C2-symmetric phosphinic acid inhibitors of HIV protease

Anusch Peyman, Karl‐Heinz Budt, Jórg Spanig et al. · Tetrahedron Letters · 1992 · 109 citations

Life Sciences, Biochemistry, Medicinal Chemistry +14

Non-peptide-based inhibitors of human immunodeficiency virus-1 protease

Anusch Peyman, Wilhelm Stahl, Konrad Wagner et al. · Bioorganic & Medicinal Chemistry Letters · 1994 · 63 citations

Life Sciences, Infectious Diseases, Medicinal Chemistry +14

Structure of HOE/BAY 793 Complexed to Human Immunodeficiency Virus (HIV‐1) Protease in Two Different Crystal Forms Structure/Function Relationship and Influence of Crystal Packing

G. Lange-Savage, Harald Berchtold, A. Liesum et al. · European Journal of Biochemistry · 1997 · 29 citations · Full text

Life Sciences, Biochemistry, Pharmacology +15

HIV protease inhibitor HOE/BAY 793, structure-activity relationships in a series of C2-symmetric diols

Karl‐Heinz Budt, Anusch Peyman, Jutta Hansen et al. · Bioorganic & Medicinal Chemistry · 1995 · 21 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11