Concepedia

The discovery of GSK221149A: A potent and selective oxytocin antagonist

John Liddle, Michael Allen, Alan D. Borthwick, David P. Brooks, David E. Davies, Richard M. Edwards, Anne M. Exall, C. Hamlett, Wendy R. Irving, Andrew M. Mason,

Bioorganic & Medicinal Chemistry Letters · 2007 · 92 citations · 10 references

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10

Oxytocin receptors in the human uterus during pregnancy and parturition

Anna‐Riitta Fuchs, Fritz Fuchs, Peter Husslein et al. · American Journal of Obstetrics and Gynecology · 1984 · 614 citations

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Fast Gradient HPLC Method to Determine Compounds Binding to Human Serum Albumin. Relationships with Octanol/Water and Immobilized Artificial Membrane Lipophilicity

Klára Valkó, Shenaz Nunhuck, Chris Bevan et al. · Journal of Pharmaceutical Sciences · 2003 · 331 citations

, , +12

Expression of oxytocin receptor in human pregnant myometrium.

Tadashi Kimura, Masahiko Takemura, Shogo Nomura et al. · Endocrinology · 1996 · 208 citations · Full text

, , +15

Expression of oxytocin receptor in human pregnant myometrium

Tsuyoshi Kimura · Endocrinology · 1996 · 71 citations

, , +15

2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: identification, stereochemistry and initial SAR

Paul G. Wyatt, Michael Allen, Alan D. Borthwick et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 66 citations

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