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Bioorganic & Medicinal Chemistry · 2013 · 20 citations · 24 references
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PharmacyMolecular BiologyOncologyDrug DesignDrug DiscoveryMolecular OncologyMelanoma PharmacotherapyDna Damage Response InhibitorsMelanocytic Tumor Molecular PathologyP53 Pathway Inactivation
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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays
Ji-Hu Zhang, Thomas D.Y. Chung, Kevin R. Oldenburg · SLAS DISCOVERY · 1999 · 7K citations · Full text
Pharmacy, Medicinal Chemistry, Drug Design +16
Chemical Similarity Searching
Peter Willett, John M. Barnard, Geoffrey M. Downs · Journal of Chemical Information and Computer Sciences · 1998 · 1.8K citations
Pharmacy, Chemistry, Drug Discovery +13
Recombinant Human Tumor Necrosis Factor-α: Effects on Proliferation of Normal and Transformed Cells in Vitro
Barry J. Sugarman, Bharat B. Aggarwal, Philip E. Hass et al. · Science · 1985 · 1.6K citations
Medicine, Cancer Biology, Oncology +8
Development and optimization of a binding assay for the XIAP BIR3 domain using fluorescence polarization
Zaneta Nikolovska‐Coleska, Renxiao Wang, Xueliang Fang et al. · Analytical Biochemistry · 2004 · 557 citations
Life Sciences, Biochemistry, Molecular Biology +15
Experiences in fragment-based drug discovery
Christopher W. Murray, Marcel L. Verdonk, David C. Rees · Trends in Pharmacological Sciences · 2012 · 236 citations
Pharmacy, Medicinal Chemistry, Drug Design +11