Convenient and versatile synthesis of formyl-substituted benzoxaboroles

An Antifungal Agent Inhibits an Aminoacyl-tRNA Synthetase by Trapping tRNA in the Editing Site

Fernando Rock, Weimin Mao, A. Yaremchuk et al. · Science · 2007 · 631 citations · Full text

Life Sciences, Biochemistry, Medicinal Chemistry +17

Discovery of a New Boron-Containing Antifungal Agent, 5-Fluoro-1,3-dihydro-1-hydroxy-2,1- benzoxaborole (AN2690), for the Potential Treatment of Onychomycosis

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Pharmacy, Dermatology, Medicinal Chemistry +17

Discovery and structure–activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis

Tsutomu Akama, Stephen J. Baker, Yongkang Zhang et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 210 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Enhanced Carboxylate Binding Using Urea and Amide-Based Receptors with Internal Lewis Acid Coordination:  A Cooperative Polarization Effect

Martin Patrick Hughes, Bradley D. Smith · The Journal of Organic Chemistry · 1997 · 183 citations

Pharmacy, Chemistry, Medicinal Chemistry +17

p<i>K</i>_a Values and Geometries of Secondary and Tertiary Amines Complexed to Boronic AcidsImplications for Sensor Design

Sheryl L. Wiskur, John J. Lavigne, Hassan Aït‐Haddou et al. · Organic Letters · 2001 · 179 citations

Natural Sciences, Chemical Engineering, Chemistry +15