Stereoselective transformation of pyrazinones into substituted analogues of cis-5-amino-6-oxo-2-piperidinemethanol and cis-5-amino-2-piperidinemethanol

An unidentified depressor substance in certain tissue extracts

U. S. von Euler, J. H. Gaddum · The Journal of Physiology · 1931 · 1.6K citations · Full text

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A new synthesis of substituted 2(1<i>H</i>)‐pyrazinones

J.A.J.M. Vekemans, C. POLLERS‐WIEERS, Georges J. Hoornaert · Journal of Heterocyclic Chemistry · 1983 · 91 citations

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Synthesis of a conformationally restricted dipeptide analogue and its evaluation as a β-turn mimic

Wim M. De Borggraeve, Frederik Rombouts, Erik V. Van der Eycken et al. · Tetrahedron Letters · 2001 · 32 citations

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Gem-disubstituted amino-ether based substance p antagonists

Timothy Harrison, B.J. Williams, Christopher J. Swain · Bioorganic & Medicinal Chemistry Letters · 1994 · 27 citations

Medicine, Medicinal Chemistry, Pharmacology +7

Cycloadducts of ethene with 2(1H)-pyrazinones and their conversion into 2,5-diazabicyclo[2.2.2]octane-3,6-diones.

Patrick K. Loosen, Mayoka G. Tutonda, Masoumeh F. Khorasani et al. · Tetrahedron · 1991 · 24 citations

Natural Sciences, Chemistry, Organic Chemistry +7