MedChemComm · 2015 · 11 citations · 21 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryMolecular PharmacologyLead Compound DesignPotency OptimizationReceptor PharmacologyPyrimidine AnalogsPyrimidine AnaloguesPyrimidine Chemistry
A series of 2-(pyridinyl)pyrimidines were identified as potent GPR40 antagonists.
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Lipophilicity in drug discovery
Michael J. Waring · Expert Opinion on Drug Discovery · 2010 · 844 citations
Celia P. Briscoe, Andrew J. Peat, Stephen C. McKeown et al. · British Journal of Pharmacology · 2006 · 400 citations · Full text