Concepedia

N-Benzyl-1-heteroaryl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamides as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1)

Martin Allan, Sukhdev Manku, Éric Therrien, Natalie Nguyen, Sylvia Styhler, Marie‐France Robert, Anne-Christine Goulet, Andrea J. Petschner, Gabi Rahil, A. Robert MacLeod,

Bioorganic & Medicinal Chemistry Letters · 2008 · 87 citations · 34 references

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References

34

Regulation of Transcription by a Protein Methyltransferase

Dagang Chen, Han Ma, Heng Hong et al. · Science · 1999 · 1.2K citations

, , +17

Ordered Cooperative Functions of PRMT1, p300, and CARM1 in Transcriptional Activation by p53

Woojin An, Jaehoon Kim, Robert G. Roeder · Cell · 2004 · 500 citations · Full text

, , +13

A Transcriptional Switch Mediated by Cofactor Methylation

Wei Xu, Hong-Wu Chen, Keyong Du et al. · Science · 2001 · 406 citations

, , +17

The Arginine Methyltransferase CARM1 Regulates the Coupling of Transcription and mRNA Processing

Donghang Cheng, Jocelyn Côté, Salam Shaaban et al. · Molecular Cell · 2007 · 381 citations · Full text

, , +14

A Novel Cell Line, MDA-kb2, That Stably Expresses an Androgen- and Glucocorticoid-Responsive Reporter for the Detection of Hormone Receptor Agonists and Antagonists

Vickie S. Wilson · Toxicological Sciences · 2002 · 332 citations

, , +17