Andrea J. Petschner

N-Benzyl-1-heteroaryl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamides as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1)

Martin Allan, Sukhdev Manku, Éric Therrien et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 87 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +7

Constrained (l-)-S-adenosyl-l-homocysteine (SAH) analogues as DNA methyltransferase inhibitors

Ljubomir Isakovic, Oscar M. Saavedra, David B. Llewellyn et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 53 citations · Full text

Pharmacy, Medicinal Chemistry, Molecular Biology +8

SAR around (l)-S-adenosyl-l-homocysteine, an inhibitor of human DNA methyltransferase (DNMT) enzymes

Oscar M. Saavedra, Ljubomir Isakovic, David B. Llewellyn et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 49 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +8

Sulfamides as novel histone deacetylase inhibitors

Amal Wahhab, David Smil, Alain Ajamian et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 30 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +10

Synthesis and evaluation of lysine derived sulfamides as histone deacetylase inhibitors

Sukhdev Manku, Martin Allan, Natalie Nguyen et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 21 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +12