Concepedia

Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist

Timothy A. Esbenshade, Gerard B. Fox, Kathleen M. Krueger, John L. Baranowski, Thomas R. Miller, Chae Hee Kang, Lynne Denny, David G. Witte, Betty Yao, Jia Bao Pan,

Biochemical Pharmacology · 2004 · 68 citations · 44 references

DOI

Concepts

References

44

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

, , +14

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 902 citations

, , +15

pA, A NEW SCALE FOR THE MEASUREMENT OF DRUG ANTAGONISM

H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1947 · 759 citations · Full text

, , +10

Cloning and Functional Expression of the Human Histamine H<sub>3</sub>Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

, , +16